Active ingredientVorapaxar SulfateCat. No. P-V060-001CAS 705260-08-8
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Stable isotope labelled · Vorapaxar family
Pharmaceutical analytical standardVorapaxar-d5
- Cat. No.
- P-V060-002
- CAS
- N/A
- Alternative CAS
- N/A
- Formula
- C29H28D5FN2O4
- Molecular weight
- 497.62 g/mol
- Category
- Stable isotope labelled
Family: Vorapaxar
An antiplatelet drug that blocks the PAR-1 receptor, through which thrombin activates platelets; approved in the United States in 2014 to reduce the risk of cardiovascular events in people who have had a heart attack or have peripheral arterial disease.
Did you know?It is derived from himbacine, an alkaloid of the tropical tree Galbulimima belgraveana, found from Queensland to New Guinea and the Solomon Islands; it has an unusually long half-life, 5 to 13 days.
The two levels compared
| Level 1 Mass balance | Level 2 Mass balance + qNMR | |
|---|---|---|
| Identity (IR, MS, 1H and 13C-NMR; peptides: ESI-MS, MALDI-TOF and IR) | ✓ | ✓ |
| HPLC purity (min. 95%) | ✓ | ✓ |
| Content by mass balance (min. 90%; peptides: for information only)* | ✓ | ✓ |
| Content verified by qNMR (small molecules only) | · | ✓ |
| Suitable to qualify it as an in-house primary standard (ICH Q7) | · | ✓ |
* Mass balance is performed on every molecule. The only exceptions are cases where the chemistry of the molecule prevents it, for example oils and highly volatile substances, on which some of the required measurements cannot be made: in those cases the CoA states how the content was assigned.
What you receive
The analytical standard
Shipped under controlled temperature when the molecule requires it.
Certificate of analysis (CoA)
For every lot: identity, purity and assay, with the supporting spectra and chromatograms.
Safety data sheet (SDS)
Sent with every order.
Tracked shipment
Follow your shipment live, from our warehouse to your lab.
More products in the Vorapaxar family
Active ingredientVorapaxar SulfateCat. No. P-V060-001CAS 705260-08-8
ImpurityVorapaxar Impurity 1Cat. No. P-V060-003Frequently asked questions
Is mass balance always performed?
Yes, on every molecule. The only exceptions are cases where the chemistry of the molecule prevents it: for example oils and highly volatile substances, on which some measurements (such as thermogravimetry) cannot be made. In those cases the CoA states which method was used to assign the content.
Can I ask for a different quantity?
Yes. The quantities are only suggestions: choose "Other" and enter the milligrams or grams you need.
Which level should I choose?
Level 1 is enough for most routine testing. Level 2 adds an independent qNMR content value and is meant for labs that need to qualify an in-house primary standard. For peptides and similar molecules, Level 2 is not available.
When will I get the quote?
Within 24 working hours, with price, availability and delivery time.
Need a molecule you cannot find?
Custom synthesis of impurities, metabolites and labelled compounds, with the same characterisation level.